http://www.cnr.it/ontology/cnr/individuo/unitaDiPersonaleInterno/MATRICOLA8061
LEONARDO PIERPAOLO MANZONI
- Type
- Label
- LEONARDO PIERPAOLO MANZONI (literal)
- LEONARDO PIERPAOLO MANZONI (literal)
- Gestore di
- Partecipa a commessa
- Persona in rapporto
- Autore CNR di
- Cyclic RGD Functionalized Gold Nanoparticles for Tumor Targeting (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Integrin-Mediated Drug Delivery in Cancer and Cardiovascular Diseases with Peptide-Functionalized Nanoparticles (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Computational design of novel peptidomimetic inhibitors of cadherin homophilic interactions (Articolo in rivista) (Prodotto della ricerca)
- Functionalized Cyclic RGD Peptidomimetics: Conjugable ligands for alpha(v)beta(3) Receptor Imaging (Articolo in rivista) (Prodotto della ricerca)
- Structural Basis for Bivalent Smac-Mimetics Recognition in the IAP Protein Family (Articolo in rivista) (Prodotto della ricerca)
- Stereoselective synthesis of C-alpha-tetrasubstituted azabicyclo[X.3.0]alkane amino acids (Articolo in rivista) (Prodotto della ricerca)
- Preparation of peptidomimetic azabicycloalkane compounds containing the RGD sequence for use as integrin inhibitors (Brevetto) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1601)
- Characterization of iron oxide-gold core-shell multifunctional nanoparticles in biomedical imaging (Contributo in atti di convegno) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1301)
- Stereoselective synthesis of peptidomimetic compounds as intermediates in the preparation of integrin antagonists (Brevetto) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1601)
- Synthesis of Gd and (68) Ga Complexes in Conjugation with a Conformationally Optimized RGD Sequence as Potential MRI and PET Tumor-Imaging Probes (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Practical stereoselective synthesis of conformationally constrained unnatural proline-based amino acids and peptidomimetics (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Preparation of peptidomimetics as integrino inhibitors (Brevetto) (Prodotto della ricerca)
- Design, synthesis, conformational analysis and application of azabicycloalkane amino acids as constrained dipeptide mimics (Articolo in rivista) (Prodotto della ricerca)
- Nonpeptide Integrin Antagonists: RGD Mimetics Incorporating Substituted Azabicycloalkanes as Amino Acid Replacements (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Rapid synthesis of oligosaccharides using an anomeric fluorous silyl protective group (Articolo in rivista) (Prodotto della ricerca)
- Targeting the X-Linked Inhibitor of Apoptosis Protein through 4-Substituted Azabicyclo[5.3.0]alkane Smac Mimetics. Structure, Activity, and Recognition Principles (Articolo in rivista) (Prodotto della ricerca)
- Mimics of Ganglioside GM1 as Cholera Toxin Ligands: Replacement of the GalNAC Residue (Articolo in rivista) (Prodotto della ricerca)
- Molecular targeting of imaging and drug delivery probes in Atherosclerosis (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- New SMAC mimetic compounds as apoptosis inducers (Brevetto) (Prodotto della ricerca)
- Enhancement of the Uptake and Cytotoxic Activity of Doxorubicin in Cancer Cells by Novel cRGD-Semipeptide-Anchoring Liposomes (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Cyclic RGD-Peptidomimetics Containing Bifunctional Diketopiperazine Scaffolds as New Potent Integrin Ligands (Articolo in rivista) (Prodotto della ricerca)
- Designing Smac-mimetics as antagonists of XIAP, cIAP1, and cIAP2 (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis of functionalized azabicycloalkane amino acids as dipeptide mimics (Articolo in rivista) (Prodotto della ricerca)
- A Potent Integrin Antagonist from a Small Library of Cyclic RGD Pentapeptide Mimics Including Benzyl-Substituted Azabicycloalkane Amino Acids (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis of the Lewis a trisaccharide based on an anomeric silyl fuorous tag (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Click chemistry to functionalise peptidomimetics (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Biological and molecular properties of a new avb3/avb5 integrin antagonist (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis and biological evaluation of dual action cyclo-RGD/SMAC mimetic conjugates targeting alphavbeta3/alphavbeta5 integrins and IAP proteins (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Potent Integrin Antagonists from a Small Library of RGD-Including Cyclic Pseudopeptides (Articolo in rivista) (Prodotto della ricerca)
- Synthesis of conformationally restricted and optically pure analogues of serine-proline dipeptide via aldolic condensation (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis of some oligopyridine-galactose conjugates and their metal complexes: a simple entry to multivalent sugar ligands (Articolo in rivista) (Prodotto della ricerca)
- Functionalised azabicycloalkane amino acids by nitrone 1,3-dipolar intramolecular cycloaddition (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Integrin targeted cyclopeptide ligands, their preparation and use (Brevetto) (Prodotto della ricerca)
- Integrin targeted synthetic ligands for diagnostic and therapeutic applications (Brevetto) (Prodotto della ricerca)
- MicroPET/CT imaging of alphavbeta3 integrin via a novel 68Ga-NOTA-RGD peptidomimetic conjugate in rat myocardial infarction (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Stereoselective synthesis of a functionalized 2-oxo-1-azabicyclo[5.3.0]alkane as a potential scaffold for targeted chemotherapy strategieseted chemoterapy strategies (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis of substituted conformationally constrained 6,5- and 7,5-fused bicyclic lactams as dipeptide mimics (Articolo in rivista) (Prodotto della ricerca)
- Froc: A New Fluorous Protective Group for Peptide and Oligosaccharide Synthesis (Articolo in rivista) (Prodotto della ricerca)
- The first example of ring-closing metathesis of dehydroamino acids: an application to the synthesis of azabicyclo[X.Y.0]alkanes (Articolo in rivista) (Prodotto della ricerca)
- Targeting integrins: insights into structure and activity of cyclic RGD pentapeptide mimics containing azabicycloalkane amino acids (Articolo in rivista) (Prodotto della ricerca)
- Iron oxide-gold core-shell nanoparticles as multimodal imaging contrast agent (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis of new bicyclic lactam petptidomimetics by ring-closing metathesis reactions (Articolo in rivista) (Prodotto della ricerca)
- Peptidomimetic compounds and preparation of biologically active derivatives (Brevetto) (Brevetto)
- Synthesis of compounds with biological activity (Brevetto) (Brevetto)
- Design, Synthesis, and Biological Evaluation of Novel cRGD- Paclitaxel Conjugates for Integrin-Assisted Drug Delivery (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- A new optical imaging probe targeting alphaVbeta3 integrin in glioblastoma xenografts (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Novel second mitochondria-derived activator of caspases (Smac) mimetic compounds sensitize human leukemic cell lines to conventional chemotherapeutic drug-induced and death receptor-mediated apoptosis (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Linkers nella sintesi organica in fase solida (Comunicazione a convegno) (Prodotto della ricerca)
- Dimeric Smac mimetics/IAP inhibitors as in vivo-active pro-apoptotic agents. Part II: Structural and biological characterization. (Articolo in rivista) (Prodotto della ricerca)
- Homo- and heterodimeric Smac mimetics/IAP inhibitors as in vivo-active pro-apoptotic agents. Part I: Synthesis (Articolo in rivista) (Prodotto della ricerca)
- 4-Aminoproline-based arginine-glycine-aspartate integrin binders with exposed ligation points: practical in-solution synthesis, conjugation and binding affinity evaluation (Articolo in rivista) (Prodotto della ricerca)
- Novel SMAC-mimetics synergistically stimulate melanoma cell death in combination with TRAIL and Bortezomib (Articolo in rivista) (Prodotto della ricerca)
- Rational design, synthesis and characterization of potent, non-peptidic Smac mimics/XIAP inhibitors as proapoptotic agents for cancer therapy (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Cyclic RGD-Containing Functionalized Azabicycloalkane Peptides as Potent Integrin Antagonists for Tumor Targeting (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Coautore
- Responsabile di
- Nome
- LEONARDO PIERPAOLO (literal)
- Cognome
- Afferisce a
- Ha pubblicazioni con
Incoming links:
- Ha afferente
- Responsabile
- Coautore
- Partecipazione di
- Ha pubblicazioni con
- Gestore
- Rapporto con persona
- Autore CNR
- Mimics of Ganglioside GM1 as Cholera Toxin Ligands: Replacement of the GalNAC Residue (Articolo in rivista) (Prodotto della ricerca)
- Rapid synthesis of oligosaccharides using an anomeric fluorous silyl protective group (Articolo in rivista) (Prodotto della ricerca)
- The first example of ring-closing metathesis of dehydroamino acids: an application to the synthesis of azabicyclo[X.Y.0]alkanes (Articolo in rivista) (Prodotto della ricerca)
- A Potent Integrin Antagonist from a Small Library of Cyclic RGD Pentapeptide Mimics Including Benzyl-Substituted Azabicycloalkane Amino Acids (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Designing Smac-mimetics as antagonists of XIAP, cIAP1, and cIAP2 (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Cyclic RGD-Peptidomimetics Containing Bifunctional Diketopiperazine Scaffolds as New Potent Integrin Ligands (Articolo in rivista) (Prodotto della ricerca)
- Synthesis of substituted conformationally constrained 6,5- and 7,5-fused bicyclic lactams as dipeptide mimics (Articolo in rivista) (Prodotto della ricerca)
- Stereoselective synthesis of a functionalized 2-oxo-1-azabicyclo[5.3.0]alkane as a potential scaffold for targeted chemotherapy strategieseted chemoterapy strategies (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Potent Integrin Antagonists from a Small Library of RGD-Including Cyclic Pseudopeptides (Articolo in rivista) (Prodotto della ricerca)
- Biological and molecular properties of a new avb3/avb5 integrin antagonist (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Click chemistry to functionalise peptidomimetics (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis of functionalized azabicycloalkane amino acids as dipeptide mimics (Articolo in rivista) (Prodotto della ricerca)
- Design, synthesis, conformational analysis and application of azabicycloalkane amino acids as constrained dipeptide mimics (Articolo in rivista) (Prodotto della ricerca)
- Stereoselective synthesis of C-alpha-tetrasubstituted azabicyclo[X.3.0]alkane amino acids (Articolo in rivista) (Prodotto della ricerca)
- Rational design, synthesis and characterization of potent, non-peptidic Smac mimics/XIAP inhibitors as proapoptotic agents for cancer therapy (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Cyclic RGD-Containing Functionalized Azabicycloalkane Peptides as Potent Integrin Antagonists for Tumor Targeting (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Novel second mitochondria-derived activator of caspases (Smac) mimetic compounds sensitize human leukemic cell lines to conventional chemotherapeutic drug-induced and death receptor-mediated apoptosis (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- A new optical imaging probe targeting alphaVbeta3 integrin in glioblastoma xenografts (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis of new bicyclic lactam petptidomimetics by ring-closing metathesis reactions (Articolo in rivista) (Prodotto della ricerca)
- Targeting integrins: insights into structure and activity of cyclic RGD pentapeptide mimics containing azabicycloalkane amino acids (Articolo in rivista) (Prodotto della ricerca)
- Froc: A New Fluorous Protective Group for Peptide and Oligosaccharide Synthesis (Articolo in rivista) (Prodotto della ricerca)
- Functionalised azabicycloalkane amino acids by nitrone 1,3-dipolar intramolecular cycloaddition (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis of some oligopyridine-galactose conjugates and their metal complexes: a simple entry to multivalent sugar ligands (Articolo in rivista) (Prodotto della ricerca)
- Synthesis of conformationally restricted and optically pure analogues of serine-proline dipeptide via aldolic condensation (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis of the Lewis a trisaccharide based on an anomeric silyl fuorous tag (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Nonpeptide Integrin Antagonists: RGD Mimetics Incorporating Substituted Azabicycloalkanes as Amino Acid Replacements (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Structural Basis for Bivalent Smac-Mimetics Recognition in the IAP Protein Family (Articolo in rivista) (Prodotto della ricerca)
- Functionalized Cyclic RGD Peptidomimetics: Conjugable ligands for alpha(v)beta(3) Receptor Imaging (Articolo in rivista) (Prodotto della ricerca)
- Cyclic RGD Functionalized Gold Nanoparticles for Tumor Targeting (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Linkers nella sintesi organica in fase solida (Comunicazione a convegno) (Prodotto della ricerca)
- Preparation of peptidomimetics as integrino inhibitors (Brevetto) (Prodotto della ricerca)
- Stereoselective synthesis of peptidomimetic compounds as intermediates in the preparation of integrin antagonists (Brevetto) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1601)
- Synthesis of compounds with biological activity (Brevetto) (Brevetto)
- Peptidomimetic compounds and preparation of biologically active derivatives (Brevetto) (Brevetto)
- Preparation of peptidomimetic azabicycloalkane compounds containing the RGD sequence for use as integrin inhibitors (Brevetto) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1601)
- Targeting the X-Linked Inhibitor of Apoptosis Protein through 4-Substituted Azabicyclo[5.3.0]alkane Smac Mimetics. Structure, Activity, and Recognition Principles (Articolo in rivista) (Prodotto della ricerca)
- Novel SMAC-mimetics synergistically stimulate melanoma cell death in combination with TRAIL and Bortezomib (Articolo in rivista) (Prodotto della ricerca)
- New SMAC mimetic compounds as apoptosis inducers (Brevetto) (Prodotto della ricerca)
- Design, Synthesis, and Biological Evaluation of Novel cRGD- Paclitaxel Conjugates for Integrin-Assisted Drug Delivery (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Characterization of iron oxide-gold core-shell multifunctional nanoparticles in biomedical imaging (Contributo in atti di convegno) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1301)
- Synthesis of Gd and (68) Ga Complexes in Conjugation with a Conformationally Optimized RGD Sequence as Potential MRI and PET Tumor-Imaging Probes (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Practical stereoselective synthesis of conformationally constrained unnatural proline-based amino acids and peptidomimetics (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Integrin-Mediated Drug Delivery in Cancer and Cardiovascular Diseases with Peptide-Functionalized Nanoparticles (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Integrin targeted cyclopeptide ligands, their preparation and use (Brevetto) (Prodotto della ricerca)
- Integrin targeted synthetic ligands for diagnostic and therapeutic applications (Brevetto) (Prodotto della ricerca)
- 4-Aminoproline-based arginine-glycine-aspartate integrin binders with exposed ligation points: practical in-solution synthesis, conjugation and binding affinity evaluation (Articolo in rivista) (Prodotto della ricerca)
- Homo- and heterodimeric Smac mimetics/IAP inhibitors as in vivo-active pro-apoptotic agents. Part I: Synthesis (Articolo in rivista) (Prodotto della ricerca)
- Dimeric Smac mimetics/IAP inhibitors as in vivo-active pro-apoptotic agents. Part II: Structural and biological characterization. (Articolo in rivista) (Prodotto della ricerca)
- Iron oxide-gold core-shell nanoparticles as multimodal imaging contrast agent (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- MicroPET/CT imaging of alphavbeta3 integrin via a novel 68Ga-NOTA-RGD peptidomimetic conjugate in rat myocardial infarction (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Molecular targeting of imaging and drug delivery probes in Atherosclerosis (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis and biological evaluation of dual action cyclo-RGD/SMAC mimetic conjugates targeting alphavbeta3/alphavbeta5 integrins and IAP proteins (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Enhancement of the Uptake and Cytotoxic Activity of Doxorubicin in Cancer Cells by Novel cRGD-Semipeptide-Anchoring Liposomes (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Computational design of novel peptidomimetic inhibitors of cadherin homophilic interactions (Articolo in rivista) (Prodotto della ricerca)